CN Patent
CN101123878A — 氨基酸前药
Assigned to Signature R&D Holdings LLC · Expires 2008-02-13 · 18y expired
What this patent protects
本发明涉及一种前药,其包括连接到药剂或药物的氨基酸,所述药剂或药物上具有羟基、氨基、羧基或其酰化衍生物。所述前药可与制备前药的药物一样使用,但治疗性能增强了。事实上,本发明的前药增强了至少两个治疗性能,如所定义的。本发明还涉及含有前药的药物组合物。
USPTO Abstract
本发明涉及一种前药,其包括连接到药剂或药物的氨基酸,所述药剂或药物上具有羟基、氨基、羧基或其酰化衍生物。所述前药可与制备前药的药物一样使用,但治疗性能增强了。事实上,本发明的前药增强了至少两个治疗性能,如所定义的。本发明还涉及含有前药的药物组合物。
Drugs covered by this patent
- Abilify (aripiprazole) · Generic (originally Otsuka/BMS)
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.