CA3027840C — Method for producing substituted polycyclic pyridone derivative and crystal of same
Assigned to Shionogi and Co Ltd · Expires 2025-09-23 · 1y expired
What this patent protects
Provided is a method for producing a substituted polycyclic pyridone derivative. A method for producing a compound represented by formula (II), which is characterized in that a compound represented by formula (I) is reacted with a compound represented by formula R2-OH (wherein R2…
USPTO Abstract
Provided is a method for producing a substituted polycyclic pyridone derivative. A method for producing a compound represented by formula (II), which is characterized in that a compound represented by formula (I) is reacted with a compound represented by formula R2-OH (wherein R2 represents an unsubstituted alkyl group) in the presence of a sodium salt and/or a magnesium salt. (In formula (I), R1 represents a hydrogen atom or a protecting group other than an unsubstituted alkyl group.) (In formula (II), R2 is as defined above.)
Drugs covered by this patent
- Xofluza (BALOXAVIR MARBOXIL) · Roche
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.