AU2020378025A1 — Crystal form of Aprocitentan, preparation method therefor and use thereof
Assigned to Crystal Pharmaceutical Suzhou Co Ltd · Expires 2022-06-23 · 4y expired
What this patent protects
Disclosed are a new crystal form of Aprocitentan (referred to as "Compound I"), a preparation method therefor, a pharmaceutical composition comprising the crystal form, and the use of the crystal form in the preparation of dual endothelin receptor antagonist drugs and dru…
USPTO Abstract
Disclosed are a new crystal form of Aprocitentan (referred to as "Compound I"), a preparation method therefor, a pharmaceutical composition comprising the crystal form, and the use of the crystal form in the preparation of dual endothelin receptor antagonist drugs and drugs for the treatment of refractory hypertension. The crystal form of Aprocitentan provided has one or more improved properties, which is of great value to the optimization and development of the drug in the future.
Drugs covered by this patent
- Tryvio (APROCITENTAN) · Idorsia
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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