AU2018278844A1 — 19-Nor C3,3-Disubstituted C21-N-Pyrazolyl Steroids And Methods Of Use Thereof
Assigned to Sage Therapeutics LLC · Expires 2019-01-03 · 7y expired
What this patent protects
Provided herein are 19-nor C3,3-disubstituted C21 -pyrazolyl steroids of Formula (I): R3R3b 21 H011.- 3 1 5 6 R4b R1 R 4a and pharmaceutically acceptable salts thereof; wherein-, R', R2, R3a, R3b, R4a, R4b, R , R6 , and R7are as defined herein. Such compounds are contemplated use…
USPTO Abstract
Provided herein are 19-nor C3,3-disubstituted C21 -pyrazolyl steroids of Formula (I): R3R3b 21 H011.- 3 1 5 6 R4b R1 R 4a and pharmaceutically acceptable salts thereof; wherein-, R', R2, R3a, R3b, R4a, R4b, R , R6 , and R7are as defined herein. Such compounds are contemplated useful for the prevention and treatment of a variety of CNS-related conditions, for example, treatment of sleep disorders, mood disorders, schizophrenia spectrum disorders, convulsive disorders, disorders of memory and/or cognition, movement disorders, personality disorders, autism spectrum disorders, pain, traumatic brain injury, vascular diseases, substance abuse disorders and/or withdrawal syndromes, and tinnitus.
Drugs covered by this patent
- Zurzuvae (ZURANOLONE) · Biogen
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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