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Ziv aflibercept
Ziv aflibercept is a VEGF inhibitor / Antiangiogenic agent Small molecule drug developed by Marashi Eye Clinic. It is currently FDA-approved for Retinal vein occlusion (RVO) with macular edema, Diabetic macular edema (DME), Age-related macular degeneration (AMD). Also known as: ZALTRAP.
Ziv-aflibercept is a recombinant fusion protein that acts as a soluble decoy receptor, binding and sequestering vascular endothelial growth factor (VEGF) and placental growth factor (PlGF) to inhibit neovascularization.
Ziv-aflibercept is a recombinant fusion protein that acts as a soluble decoy receptor, binding and sequestering vascular endothelial growth factor (VEGF) and placental growth factor (PlGF) to inhibit neovascularization. Used for Retinal vein occlusion (RVO) with macular edema, Diabetic macular edema (DME), Age-related macular degeneration (AMD).
At a glance
| Generic name | Ziv aflibercept |
|---|---|
| Also known as | ZALTRAP |
| Sponsor | Marashi Eye Clinic |
| Drug class | VEGF inhibitor / Antiangiogenic agent |
| Target | VEGF-A, VEGF-B, PlGF (Placental Growth Factor) |
| Modality | Small molecule |
| Therapeutic area | Ophthalmology |
| Phase | FDA-approved |
Mechanism of action
Ziv-aflibercept functions as a VEGF trap by combining the extracellular domains of VEGF receptors 1 and 2 fused to the Fc portion of human immunoglobulin G1. This construct binds circulating VEGF and PlGF with high affinity, preventing their interaction with endogenous receptors on endothelial cells and thereby suppressing pathological angiogenesis. It is administered as an intravitreal injection for ocular neovascular diseases.
Approved indications
- Retinal vein occlusion (RVO) with macular edema
- Diabetic macular edema (DME)
- Age-related macular degeneration (AMD)
Common side effects
- Conjunctival hemorrhage
- Eye pain
- Floaters
- Intraocular pressure elevation
- Endophthalmitis
Key clinical trials
- Testing the PD-1 Antibody, MK3475, Given With Ziv-aflibercept in Patients With Advanced Cancer (PHASE1)
- A Clinical Trial of EYE201/MK-8748 in People With Macular Degeneration (MK-8748-003) (PHASE2, PHASE3)
- Extension Study to Evaluate the Long-Term Outcomes of Pediatric Patients Who Received Treatment for Retinopathy of Prematurity in the VGFTe-ROP-1920 Study (Acronym: Butterfleye Next)
- 4D-150 in Patients With Macular Neovascularization Secondary to Age-Related Macular Degeneration (PHASE3)
- A Clinical Study of QL1207H Injection Versus Aflibercept for Neovascular Age-related Macular Degeneration (PHASE3)
- Clinical Study to Compare Efficacy and Safety of AVT29 and Eylea HD in Participants With Diabetic Macular Edema (PHASE3)
- Efficacy and Safety Study of Ixoberogene Soroparvovec (Ixo-vec) in Participants With Neovascular Age-related Macular Degeneration (AQUARIUS) (PHASE3)
- An Observational Study to Collect Data on How Aflibercept (Eylea) Given Using a Paediatric Dosing Device is Used in Preterm Babies With Retinopathy of Prematurity in the United Kingdom (UK)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Ziv aflibercept CI brief — competitive landscape report
- Ziv aflibercept updates RSS · CI watch RSS
- Marashi Eye Clinic portfolio CI
Frequently asked questions about Ziv aflibercept
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Related
- Drug class: All VEGF inhibitor / Antiangiogenic agent drugs
- Target: All drugs targeting VEGF-A, VEGF-B, PlGF (Placental Growth Factor)
- Manufacturer: Marashi Eye Clinic — full pipeline
- Therapeutic area: All drugs in Ophthalmology
- Indication: Drugs for Retinal vein occlusion (RVO) with macular edema
- Indication: Drugs for Diabetic macular edema (DME)
- Indication: Drugs for Age-related macular degeneration (AMD)
- Also known as: ZALTRAP
- Compare: Ziv aflibercept vs similar drugs
- Pricing: Ziv aflibercept cost, discount & access