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Vitamin D3 tablets

Ain Shams University · FDA-approved active Small molecule

Vitamin D3 acts as a hormone precursor that is converted in the body to its active form, calcitriol, which regulates calcium and phosphate homeostasis and modulates immune function.

Vitamin D3 acts as a hormone precursor that is converted in the body to its active form, calcitriol, which regulates calcium and phosphate homeostasis and modulates immune function. Used for Vitamin D deficiency prevention and treatment, Osteoporosis and bone health support, Calcium absorption enhancement.

At a glance

Generic nameVitamin D3 tablets
Also known asVigantoletten, Vigantoletten; Merck Pharma, Germany
SponsorAin Shams University
Drug classVitamin D supplement / Secosteroid
TargetVitamin D receptor (VDR)
ModalitySmall molecule
Therapeutic areaNutritional supplementation / Bone health / Immunology
PhaseFDA-approved

Mechanism of action

Vitamin D3 (cholecalciferol) is hydroxylated in the liver to 25-hydroxyvitamin D and then in the kidneys to the active metabolite 1,25-dihydroxyvitamin D (calcitriol). Calcitriol binds to the vitamin D receptor (VDR) in target tissues, promoting intestinal calcium and phosphate absorption, bone mineralization, and immune cell differentiation. It also has pleiotropic effects on cell proliferation, differentiation, and immune regulation.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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