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Vitamin D3 (High dose)

Shiraz University of Medical Sciences · Phase 3 active Small molecule

High-dose vitamin D3 acts as a ligand for the vitamin D receptor to regulate calcium and phosphate homeostasis, immune function, and cellular differentiation.

High-dose vitamin D3 acts as a ligand for the vitamin D receptor to regulate calcium and phosphate homeostasis, immune function, and cellular differentiation. Used for COVID-19 (phase 3 trial context), Vitamin D deficiency.

At a glance

Generic nameVitamin D3 (High dose)
Also known ascholecalciferol
SponsorShiraz University of Medical Sciences
Drug classVitamin D analog / Secosteroid
TargetVitamin D receptor (VDR)
ModalitySmall molecule
Therapeutic areaImmunology / Infectious Disease / Bone Metabolism
PhasePhase 3

Mechanism of action

Vitamin D3 (cholecalciferol) binds to the vitamin D receptor (VDR) in target tissues, modulating the expression of genes involved in calcium absorption, bone metabolism, and immune regulation. At high doses, it may exert immunomodulatory and anti-inflammatory effects beyond classical calcium homeostasis, potentially beneficial in conditions with dysregulated immune responses or chronic inflammation.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results