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Vincristine + Carboplatin + Etoposide

St. Jude Children's Research Hospital · Phase 3 active Small molecule

Vincristine + Carboplatin + Etoposide is a Vinca alkaloid, platinum-based alkylating agent, topoisomerase inhibitor Small molecule drug developed by St. Jude Children's Research Hospital. It is currently in Phase 3 development for Small cell lung cancer, Non-small cell lung cancer, Hodgkin lymphoma. Also known as: Oncovin + Paraplatin + VP-16.

Vincristine is a vinca alkaloid that inhibits microtubule formation, disrupting cell division. Carboplatin is a platinum-based alkylating agent that cross-links DNA, causing cell death. Etoposide is a topoisomerase inhibitor that prevents DNA replication and transcription.

Vincristine is a vinca alkaloid that inhibits microtubule formation, disrupting cell division. Carboplatin is a platinum-based alkylating agent that cross-links DNA, causing cell death. Etoposide is a topoisomerase inhibitor that prevents DNA replication and transcription. Used for Small cell lung cancer, Non-small cell lung cancer, Hodgkin lymphoma.

At a glance

Generic nameVincristine + Carboplatin + Etoposide
Also known asOncovin + Paraplatin + VP-16
SponsorSt. Jude Children's Research Hospital
Drug classVinca alkaloid, platinum-based alkylating agent, topoisomerase inhibitor
TargetMicrotubules, DNA
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

Vincristine works by binding to tubulin and preventing the formation of microtubules, which are essential for cell division. This leads to cell cycle arrest and apoptosis. Carboplatin, on the other hand, forms platinum-DNA adducts that interfere with DNA replication and transcription, ultimately causing cell death. Etoposide inhibits topoisomerase II, an enzyme that unwinds DNA during replication and transcription, leading to DNA damage and cell death.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Vincristine + Carboplatin + Etoposide

What is Vincristine + Carboplatin + Etoposide?

Vincristine + Carboplatin + Etoposide is a Vinca alkaloid, platinum-based alkylating agent, topoisomerase inhibitor drug developed by St. Jude Children's Research Hospital, indicated for Small cell lung cancer, Non-small cell lung cancer, Hodgkin lymphoma.

How does Vincristine + Carboplatin + Etoposide work?

Vincristine is a vinca alkaloid that inhibits microtubule formation, disrupting cell division. Carboplatin is a platinum-based alkylating agent that cross-links DNA, causing cell death. Etoposide is a topoisomerase inhibitor that prevents DNA replication and transcription.

What is Vincristine + Carboplatin + Etoposide used for?

Vincristine + Carboplatin + Etoposide is indicated for Small cell lung cancer, Non-small cell lung cancer, Hodgkin lymphoma, Testicular cancer.

Who makes Vincristine + Carboplatin + Etoposide?

Vincristine + Carboplatin + Etoposide is developed by St. Jude Children's Research Hospital (see full St. Jude Children's Research Hospital pipeline at /company/st-jude-children-s-research-hospital).

Is Vincristine + Carboplatin + Etoposide also known as anything else?

Vincristine + Carboplatin + Etoposide is also known as Oncovin + Paraplatin + VP-16.

What drug class is Vincristine + Carboplatin + Etoposide in?

Vincristine + Carboplatin + Etoposide belongs to the Vinca alkaloid, platinum-based alkylating agent, topoisomerase inhibitor class. See all Vinca alkaloid, platinum-based alkylating agent, topoisomerase inhibitor drugs at /class/vinca-alkaloid-platinum-based-alkylating-agent-topoisomerase-inhibitor.

What development phase is Vincristine + Carboplatin + Etoposide in?

Vincristine + Carboplatin + Etoposide is in Phase 3.

What are the side effects of Vincristine + Carboplatin + Etoposide?

Common side effects of Vincristine + Carboplatin + Etoposide include Neutropenia, Thrombocytopenia, Anemia, Nausea and vomiting, Diarrhea, Fatigue.

What does Vincristine + Carboplatin + Etoposide target?

Vincristine + Carboplatin + Etoposide targets Microtubules, DNA and is a Vinca alkaloid, platinum-based alkylating agent, topoisomerase inhibitor.

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