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Vedolizumab SC

Takeda · FDA-approved active Small molecule

Vedolizumab is a monoclonal antibody that selectively blocks the α4β7 integrin on gut-homing lymphocytes, preventing their migration to the gastrointestinal tract.

Vedolizumab SC, developed by Takeda, is a monoclonal antibody targeting gut-specific inflammation. It is currently in Phase 3 and 4 trials for ulcerative colitis and Crohn's disease, with a strong safety profile and promising efficacy. The drug is not yet FDA-approved but has several ongoing and completed trials.

At a glance

Generic nameVedolizumab SC
Also known asMLN0002SC, MLN0002, ENTYVIO, KYNTELES, MLN0002, Entyvio, MLN0002, ENTYVIO, KYNTELES
SponsorTakeda
Drug classIntegrin antagonist; monoclonal antibody
Targetα4β7 integrin
ModalitySmall molecule
Therapeutic areaImmunology / Gastroenterology
PhaseFDA-approved

Mechanism of action

By binding to α4β7 integrin expressed on memory T cells, vedolizumab prevents these cells from adhering to mucosal addressin cell adhesion molecule-1 (MAdCAM-1) on gut endothelial cells. This blocks lymphocyte trafficking to the intestinal mucosa, reducing local inflammation in inflammatory bowel disease. The subcutaneous formulation (SC) provides an alternative to intravenous administration with improved patient convenience.

Approved indications

Common side effects

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