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Ulimorelin Invtravenously (IV)

Tranzyme, Inc. · Phase 3 active Small molecule Under review

Ulimorelin Invtravenously (IV) is a Ghrelin receptor agonist Small molecule drug developed by Tranzyme, Inc.. It is currently in Phase 3 development for Symptomatic gastroesophageal reflux disease (GERD) in patients with type 2 diabetes mellitus.

Ulimorelin is a ghrelin receptor agonist that stimulates gastric emptying.

Ulimorelin is a small molecule administered intravenously (IV) for the treatment of gastrointestinal dysmotility. It is a synthetic compound that has been studied in clinical trials, including the ULISES 008 study, to evaluate its efficacy and safety.

Likelihood of approval
58.3% vs 58.3% industry baseline
If approved by FDA: likely 2028–2030
Steps remaining: NDA/BLA submission
Confidence: High
Why this estimate
  • Baseline phase 3 → approval rate +58.3pp
    Industry-wide phase 3 drugs reach approval ~58.3% of the time (BIO/Informa 2023 industry benchmark across all therapeutic areas).
Predicted approval windows by jurisdiction (conditional on FDA approval)
Regulator Country Likely year Lag vs FDA
FDA US 2028–2030
EMA EU 2029–2031 +0.7 yr
MHRA GB 2029–2031 +0.7 yr
Health Canada CA 2029–2032 +0.9 yr
TGA AU 2029–2032 +1.2 yr
PMDA JP 2029–2032 +1.5 yr
NMPA CN 2030–2033 +2.3 yr
MFDS KR 2029–2032 +1.4 yr
CDSCO IN 2029–2033 +1.8 yr
ANVISA BR 2030–2033 +2.3 yr

Hover any row for the lag rationale. Lag estimates are reduced when the drug has FDA Breakthrough or EMA PRIME designation (sponsors file globally in parallel).

Estimate based on the BIO/Informa industry phase transition rates plus per-drug modifiers for therapeutic area, sponsor type, FDA designations, mechanism, and trial design. Per-jurisdiction lags from Tufts CSDD international approval studies. Not investment, clinical or regulatory advice. Methodology: /methodology#likelihood.

At a glance

Generic nameUlimorelin Invtravenously (IV)
SponsorTranzyme, Inc.
Drug classGhrelin receptor agonist
TargetGhrelin receptor
ModalitySmall molecule
Therapeutic areaGastrointestinal
PhasePhase 3

Mechanism of action

Ulimorelin works by activating the ghrelin receptor, which is involved in regulating gastric motility and emptying. This leads to an increase in gastric emptying, which can help alleviate symptoms of gastroparesis.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:

Frequently asked questions about Ulimorelin Invtravenously (IV)

What is Ulimorelin Invtravenously (IV)?

Ulimorelin Invtravenously (IV) is a Ghrelin receptor agonist drug developed by Tranzyme, Inc., indicated for Symptomatic gastroesophageal reflux disease (GERD) in patients with type 2 diabetes mellitus.

How does Ulimorelin Invtravenously (IV) work?

Ulimorelin is a ghrelin receptor agonist that stimulates gastric emptying.

What is Ulimorelin Invtravenously (IV) used for?

Ulimorelin Invtravenously (IV) is indicated for Symptomatic gastroesophageal reflux disease (GERD) in patients with type 2 diabetes mellitus.

Who makes Ulimorelin Invtravenously (IV)?

Ulimorelin Invtravenously (IV) is developed by Tranzyme, Inc. (see full Tranzyme, Inc. pipeline at /company/tranzyme-inc).

What drug class is Ulimorelin Invtravenously (IV) in?

Ulimorelin Invtravenously (IV) belongs to the Ghrelin receptor agonist class. See all Ghrelin receptor agonist drugs at /class/ghrelin-receptor-agonist.

What development phase is Ulimorelin Invtravenously (IV) in?

Ulimorelin Invtravenously (IV) is in Phase 3.

What are the side effects of Ulimorelin Invtravenously (IV)?

Common side effects of Ulimorelin Invtravenously (IV) include Nausea, Diarrhea, Vomiting, Abdominal pain.

What does Ulimorelin Invtravenously (IV) target?

Ulimorelin Invtravenously (IV) targets Ghrelin receptor and is a Ghrelin receptor agonist.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing