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Triamcinolone + Lidocaine

MetroHealth Medical Center · FDA-approved active Small molecule

Triamcinolone reduces inflammation via glucocorticoid receptor activation, while lidocaine provides local anesthetic effects by blocking sodium channels in nerve fibers.

Triamcinolone reduces inflammation via glucocorticoid receptor activation, while lidocaine provides local anesthetic effects by blocking sodium channels in nerve fibers. Used for Intra-articular injection for inflammatory joint conditions, Intralesional injection for inflammatory skin conditions, Local infiltration for pain and inflammation relief.

At a glance

Generic nameTriamcinolone + Lidocaine
Also known asKenalog = Triamcinolone
SponsorMetroHealth Medical Center
Drug classCorticosteroid + Local anesthetic combination
TargetGlucocorticoid receptor (triamcinolone); voltage-gated sodium channels (lidocaine)
ModalitySmall molecule
Therapeutic areaRheumatology / Pain Management / Dermatology
PhaseFDA-approved

Mechanism of action

Triamcinolone is a synthetic corticosteroid that suppresses inflammatory and immune responses by binding to glucocorticoid receptors and inhibiting pro-inflammatory cytokine production. Lidocaine is a local anesthetic that blocks voltage-gated sodium channels, preventing nerve depolarization and pain signal transmission. Together, this combination provides both anti-inflammatory and analgesic effects at the site of injection.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results