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Treatment with tirzapatide

University Medical Centre Ljubljana · FDA-approved active Small molecule

Treatment with tirzapatide is a GLP-1/GIP receptor agonist Small molecule drug developed by University Medical Centre Ljubljana. It is currently FDA-approved for Type 2 diabetes mellitus, Chronic weight management in adults with obesity or overweight.

Tirzapatide is a dual GLP-1 and GIP receptor agonist that stimulates insulin secretion and reduces glucagon levels in response to elevated blood glucose.

Tirzapatide is a dual GLP-1 and GIP receptor agonist that stimulates insulin secretion and reduces glucagon levels in response to elevated blood glucose. Used for Type 2 diabetes mellitus, Chronic weight management in adults with obesity or overweight.

At a glance

Generic nameTreatment with tirzapatide
SponsorUniversity Medical Centre Ljubljana
Drug classGLP-1/GIP receptor agonist
TargetGLP-1R, GIPR
ModalitySmall molecule
Therapeutic areaEndocrinology/Diabetes
PhaseFDA-approved

Mechanism of action

Tirzapatide activates both glucagon-like peptide-1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP) receptors, leading to glucose-dependent insulin secretion, suppression of glucagon, and delayed gastric emptying. This dual mechanism results in improved glycemic control and weight loss in patients with type 2 diabetes. The GIP component provides additional metabolic benefits beyond traditional GLP-1 monotherapy.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Treatment with tirzapatide

What is Treatment with tirzapatide?

Treatment with tirzapatide is a GLP-1/GIP receptor agonist drug developed by University Medical Centre Ljubljana, indicated for Type 2 diabetes mellitus, Chronic weight management in adults with obesity or overweight.

How does Treatment with tirzapatide work?

Tirzapatide is a dual GLP-1 and GIP receptor agonist that stimulates insulin secretion and reduces glucagon levels in response to elevated blood glucose.

What is Treatment with tirzapatide used for?

Treatment with tirzapatide is indicated for Type 2 diabetes mellitus, Chronic weight management in adults with obesity or overweight.

Who makes Treatment with tirzapatide?

Treatment with tirzapatide is developed and marketed by University Medical Centre Ljubljana (see full University Medical Centre Ljubljana pipeline at /company/university-medical-centre-ljubljana).

What drug class is Treatment with tirzapatide in?

Treatment with tirzapatide belongs to the GLP-1/GIP receptor agonist class. See all GLP-1/GIP receptor agonist drugs at /class/glp-1-gip-receptor-agonist.

What development phase is Treatment with tirzapatide in?

Treatment with tirzapatide is FDA-approved (marketed).

What are the side effects of Treatment with tirzapatide?

Common side effects of Treatment with tirzapatide include Nausea, Vomiting, Diarrhea, Constipation, Abdominal pain, Injection site reactions.

What does Treatment with tirzapatide target?

Treatment with tirzapatide targets GLP-1R, GIPR and is a GLP-1/GIP receptor agonist.

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