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topical pimecrolimus treatment

University Hospital, Ghent · FDA-approved active Small molecule

Pimecrolimus is a calcineurin inhibitor that suppresses T-cell activation and inflammatory cytokine production in the skin.

Pimecrolimus is a calcineurin inhibitor that suppresses T-cell activation and inflammatory cytokine production in the skin. Used for Atopic dermatitis (eczema), Allergic contact dermatitis, Seborrheic dermatitis.

At a glance

Generic nametopical pimecrolimus treatment
SponsorUniversity Hospital, Ghent
Drug classCalcineurin inhibitor (topical immunosuppressant)
TargetCalcineurin
ModalitySmall molecule
Therapeutic areaDermatology/Immunology
PhaseFDA-approved

Mechanism of action

Pimecrolimus binds to calcineurin and prevents its interaction with NFAT (nuclear factor of activated T cells), thereby blocking T-cell proliferation and the release of pro-inflammatory mediators. When applied topically, it reduces skin inflammation without the systemic immunosuppression associated with oral calcineurin inhibitors, making it suitable for localized inflammatory skin conditions.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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