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The midazolam ketamine group

Kasr El Aini Hospital · Phase 3 active Small molecule

Midazolam is a benzodiazepine that acts as a GABA_A receptor agonist, while ketamine is an NMDA receptor antagonist.

Midazolam is a benzodiazepine that acts as a GABA_A receptor agonist, while ketamine is an NMDA receptor antagonist. Used for Procedural sedation and anesthesia.

At a glance

Generic nameThe midazolam ketamine group
SponsorKasr El Aini Hospital
Drug classBenzodiazepine and NMDA receptor antagonist
TargetGABA_A receptor, NMDA receptor
ModalitySmall molecule
Therapeutic areaAnesthesiology
PhasePhase 3

Mechanism of action

Midazolam's mechanism of action involves binding to the GABA_A receptor, enhancing the effect of the neurotransmitter gamma-aminobutyric acid (GABA), leading to sedative, hypnotic, anxiolytic, anticonvulsant, and muscle relaxant properties. Ketamine, on the other hand, acts as an antagonist at the NMDA receptor, which is involved in the regulation of synaptic plasticity and memory formation. The combination of midazolam and ketamine may provide synergistic effects in terms of sedation and analgesia.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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