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TDF/3TC/EFV or DTG or NVP
This is a combination antiretroviral regimen containing nucleoside reverse transcriptase inhibitors (TDF/3TC), a non-nucleoside reverse transcriptase inhibitor (EFV or NVP), or an integrase strand transfer inhibitor (DTG) that blocks HIV replication by inhibiting key viral enzymes.
This is a combination antiretroviral regimen containing nucleoside reverse transcriptase inhibitors (TDF/3TC), a non-nucleoside reverse transcriptase inhibitor (EFV or NVP), or an integrase strand transfer inhibitor (DTG) that blocks HIV replication by inhibiting key viral enzymes. Used for HIV-1 infection treatment and suppression.
At a glance
| Generic name | TDF/3TC/EFV or DTG or NVP |
|---|---|
| Sponsor | MU-JHU CARE |
| Drug class | Antiretroviral combination therapy (NRTI + NNRTI or INSTI) |
| Target | HIV reverse transcriptase, HIV integrase |
| Modality | Small molecule |
| Therapeutic area | Infectious Disease / Virology |
| Phase | FDA-approved |
Mechanism of action
TDF (tenofovir) and 3TC (lamivudine) are nucleoside reverse transcriptase inhibitors that prevent HIV reverse transcriptase from converting viral RNA to DNA. EFV (efavirenz) and NVP (nevirapine) are non-nucleoside reverse transcriptase inhibitors that directly inhibit the same enzyme through a different mechanism. DTG (dolutegravir) is an integrase inhibitor that prevents viral DNA from integrating into the host genome. These agents are used in combination to suppress HIV replication and prevent resistance.
Approved indications
- HIV-1 infection treatment and suppression
Common side effects
- Nausea
- Diarrhea
- Headache
- Dizziness (EFV)
- Rash (NVP)
- Hepatotoxicity
- Lipodystrophy
- Renal impairment (TDF)
Key clinical trials
- A Study to Provide Continued Access to Study Drug to Children and Adolescents Who Have Completed Clinical Studies Involving Gilead HIV Treatments (PHASE4)
- BONE: STAR (Switching to TAF Based Anti-Retroviral Therapy) Study (PHASE4)
- Study to Evaluate Switching From a Regimen of Two Nucleos(t)Ide Reverse Transcriptase Inhibitors (NRTI) Plus a Third Agent to a Fixed Dose Combination (FDC) of Bictegravir/Emtricitabine/Tenofovir Alafenamide (B/F/TAF), in Virologically-Suppressed, HIV-1 Infected African American Participants (PHASE3)
- Study to Evaluate Switching to Elvitegravir/Cobicistat/Emtricitabine/Tenofovir Alafenamide (E/C/F/TAF) Fixed Dose Combination (FDC) in Virologically-Suppressed HIV-1 Infected Adults Harboring the Archived Isolated NRTI Resistance Mutation M184V/M184I (PHASE3)
- Switching From a Tenofovir Disoproxil Fumarate (TDF) Containing Regimen to Elvitegravir/Cobicistat/Emtricitabine/ Tenofovir Alafenamide (E/C/F/TAF) Fixed-Dose Combination (FDC) in Virologically-Suppressed, HIV-1 Infected Adults Aged ≥ 60 Years (PHASE3)
- Switch Study to Evaluate F/TAF in HIV-1 Infected Adults Who Are Virologically Suppressed on Regimens Containing ABC/3TC (PHASE3)
- Safety and Efficacy of Switching From Regimens of ABC/3TC + a 3rd Agent to E/C/F/TAF Fixed-Dose Combination (FDC) in Virologically-Suppressed HIV 1 Infected Adults (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- TDF/3TC/EFV or DTG or NVP CI brief — competitive landscape report
- TDF/3TC/EFV or DTG or NVP updates RSS · CI watch RSS
- MU-JHU CARE portfolio CI