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sublingual nitroglycerine

United States Naval Medical Center, San Diego · Phase 3 active Small molecule

Sublingual nitroglycerine works by releasing nitric oxide, which relaxes vascular smooth muscle and reduces blood pressure.

Sublingual nitroglycerine works by releasing nitric oxide, which relaxes vascular smooth muscle and reduces blood pressure. Used for Angina pectoris, Atrial fibrillation for rate control.

At a glance

Generic namesublingual nitroglycerine
Also known asNitrolingual
SponsorUnited States Naval Medical Center, San Diego
Drug classvasodilator
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 3

Mechanism of action

This leads to vasodilation and a decrease in cardiac workload, resulting in reduced myocardial oxygen demand. Nitroglycerine is a nitrate ester prodrug that is converted to nitric oxide in the body, which then activates guanylate cyclase and increases cyclic GMP levels, leading to smooth muscle relaxation.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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