Last reviewed · How we verify

stander treatment pregabalin

Hawler Medical University · FDA-approved active Small molecule

Pregabalin binds to the alpha-2-delta subunit of voltage-gated calcium channels in the central nervous system, reducing the release of excitatory neurotransmitters.

Pregabalin binds to the alpha-2-delta subunit of voltage-gated calcium channels in the central nervous system, reducing the release of excitatory neurotransmitters. Used for Neuropathic pain (diabetic peripheral neuropathy, postherpetic neuralgia, spinal cord injury), Partial-onset seizures (adjunctive therapy), Generalized anxiety disorder.

At a glance

Generic namestander treatment pregabalin
SponsorHawler Medical University
Drug classGabapentinoid; anticonvulsant; anxiolytic
TargetAlpha-2-delta subunit of voltage-gated calcium channels
ModalitySmall molecule
Therapeutic areaNeurology; Pain Management; Psychiatry
PhaseFDA-approved

Mechanism of action

By binding to presynaptic calcium channels, pregabalin decreases calcium influx and subsequently reduces the release of glutamate, noradrenaline, and substance P. This leads to reduced neuronal excitability and pain signal transmission. The drug is effective in conditions characterized by neuropathic pain and hyperexcitability of the nervous system.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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