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Standard-dose rtPA

The George Institute · Phase 3 active Small molecule

Standard-dose rtPA works by dissolving blood clots to restore blood flow to the brain.

Standard-dose rtPA is a thrombolytic agent used primarily for acute ischemic stroke. Despite no FDA label, it is widely studied in various phases of clinical trials, including nebulized administration for ARDS due to COVID-19 and combination therapies. Key trials include ENCHANTED and the Alteplase-Tenecteplase Trial Evaluation for Stroke Thrombolysis.

At a glance

Generic nameStandard-dose rtPA
Also known asActilyse
SponsorThe George Institute
Drug classThrombolytic
TargettPA
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 3

Mechanism of action

Standard-dose rtPA is a thrombolytic agent that specifically targets plasminogen activator, which breaks down blood clots. This process helps to restore blood flow to the brain, reducing the risk of further brain damage and improving outcomes in patients with acute ischemic stroke.

Approved indications

Common side effects