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Standard-dose intravenous tenecteplase

The George Institute · Phase 3 active Small molecule

Tenecteplase is a tissue plasminogen activator that works by catalyzing the conversion of plasminogen to plasmin, resulting in the breakdown of blood clots.

Tenecteplase is a tissue plasminogen activator that works by catalyzing the conversion of plasminogen to plasmin, resulting in the breakdown of blood clots. Used for Acute ischemic stroke.

At a glance

Generic nameStandard-dose intravenous tenecteplase
SponsorThe George Institute
Drug classtissue plasminogen activator
TargettPA
ModalitySmall molecule
Therapeutic areaCardiovascular
PhasePhase 3

Mechanism of action

This process is crucial for the treatment of acute ischemic stroke, as it helps to restore blood flow to the affected area of the brain. Tenecteplase is a recombinant form of tPA, which has a higher specificity and lower risk of bleeding compared to its natural counterpart.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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