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Salmeterol Fluticasone

Università degli Studi di Brescia · FDA-approved active Small molecule

Salmeterol/fluticasone is a combination inhaled corticosteroid and long-acting beta-2 agonist that reduces airway inflammation and dilates airways to improve breathing.

Salmeterol/fluticasone is a combination inhaled corticosteroid and long-acting beta-2 agonist that reduces airway inflammation and dilates airways to improve breathing. Used for Asthma maintenance therapy, Chronic obstructive pulmonary disease (COPD) maintenance therapy.

At a glance

Generic nameSalmeterol Fluticasone
Also known asSERETIDE
SponsorUniversità degli Studi di Brescia
Drug classInhaled corticosteroid/long-acting beta-2 agonist combination
TargetGlucocorticoid receptor (fluticasone); beta-2 adrenergic receptor (salmeterol)
ModalitySmall molecule
Therapeutic areaRespiratory/Pulmonology
PhaseFDA-approved

Mechanism of action

Fluticasone is a corticosteroid that suppresses inflammatory responses in the airways by binding glucocorticoid receptors, reducing mucus production and airway edema. Salmeterol is a long-acting beta-2 agonist that binds beta-2 adrenergic receptors on airway smooth muscle, causing bronchodilation and lasting 12+ hours. Together, they provide both anti-inflammatory and bronchodilatory effects for sustained asthma and COPD control.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results