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Salmeterol 50 mcg via DISKUS

GlaxoSmithKline · FDA-approved active Small molecule

Salmeterol is a long-acting beta2-adrenergic agonist that relaxes bronchial smooth muscle to improve airflow.

Salmeterol 50 mcg via DISKUS is a long-acting beta2-adrenergic agonist (LABA) developed by GlaxoSmithKline for the maintenance treatment of asthma and chronic obstructive pulmonary disease (COPD). It works by relaxing the muscles in the airways to improve breathing. Despite its effectiveness, it carries warnings about the risk of asthma-related death when used without an inhaled corticosteroid. Common side effects include upper respiratory tract infections, headache, and muscle pain. The drug has no FDA label, which may affect its market presence and regulatory status.

At a glance

Generic nameSalmeterol 50 mcg via DISKUS
SponsorGlaxoSmithKline
Drug classLong-acting beta2-adrenergic agonist (LABA)
TargetBeta2-adrenergic receptors
ModalitySmall molecule
Therapeutic areaRespiratory
PhaseFDA-approved

Mechanism of action

Salmeterol binds to and activates beta2-adrenergic receptors on bronchial smooth muscle cells, leading to the relaxation of these muscles and improved airflow.

Approved indications

Boxed warnings

Common side effects

Drug interactions

Key clinical trials

Patents

PatentExpiryType
US5541195

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results
FDA Orange BookPatents + exclusivity

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