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Saline + Propofol

Seoul National University Hospital · FDA-approved active Small molecule

Propofol dissolved in saline acts as an intravenous anesthetic by enhancing GABAergic inhibitory neurotransmission in the central nervous system.

Propofol dissolved in saline acts as an intravenous anesthetic by enhancing GABAergic inhibitory neurotransmission in the central nervous system. Used for Induction and maintenance of general anesthesia, Sedation in intensive care units, Sedation for diagnostic and therapeutic procedures.

At a glance

Generic nameSaline + Propofol
SponsorSeoul National University Hospital
Drug classGeneral anesthetic
TargetGABA-A receptor
ModalitySmall molecule
Therapeutic areaAnesthesiology
PhaseFDA-approved

Mechanism of action

Propofol is a lipophilic alkylphenol that potentiates GABA-A receptor function, leading to increased chloride ion influx and neuronal hyperpolarization. This results in rapid onset of unconsciousness and sedation. The saline vehicle serves as a sterile diluent for intravenous administration.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results