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Rasagiline mesylate plus Mirapex

Teva Neuroscience, Inc. · FDA-approved active Small molecule

Rasagiline mesylate plus Mirapex is a MAO-B inhibitor plus dopamine agonist combination Small molecule drug developed by Teva Neuroscience, Inc.. It is currently FDA-approved for Parkinson's disease.

This combination pairs a monoamine oxidase B inhibitor with a dopamine agonist to enhance dopaminergic signaling in the brain for Parkinson's disease management.

This combination pairs a monoamine oxidase B inhibitor with a dopamine agonist to enhance dopaminergic signaling in the brain for Parkinson's disease management. Used for Parkinson's disease.

At a glance

Generic nameRasagiline mesylate plus Mirapex
SponsorTeva Neuroscience, Inc.
Drug classMAO-B inhibitor plus dopamine agonist combination
TargetMonoamine oxidase B and dopamine D2/D3 receptors
ModalitySmall molecule
Therapeutic areaNeurology
PhaseFDA-approved

Mechanism of action

Rasagiline is a selective MAO-B inhibitor that prevents the breakdown of dopamine, while Mirapex (pramipexole) is a dopamine D2/D3 receptor agonist that directly stimulates dopamine receptors. Together, they increase dopamine availability and receptor activation, providing complementary symptomatic relief in Parkinson's disease by addressing both dopamine preservation and receptor stimulation.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

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Frequently asked questions about Rasagiline mesylate plus Mirapex

What is Rasagiline mesylate plus Mirapex?

Rasagiline mesylate plus Mirapex is a MAO-B inhibitor plus dopamine agonist combination drug developed by Teva Neuroscience, Inc., indicated for Parkinson's disease.

How does Rasagiline mesylate plus Mirapex work?

This combination pairs a monoamine oxidase B inhibitor with a dopamine agonist to enhance dopaminergic signaling in the brain for Parkinson's disease management.

What is Rasagiline mesylate plus Mirapex used for?

Rasagiline mesylate plus Mirapex is indicated for Parkinson's disease.

Who makes Rasagiline mesylate plus Mirapex?

Rasagiline mesylate plus Mirapex is developed and marketed by Teva Neuroscience, Inc. (see full Teva Neuroscience, Inc. pipeline at /company/teva-neuroscience-inc).

What drug class is Rasagiline mesylate plus Mirapex in?

Rasagiline mesylate plus Mirapex belongs to the MAO-B inhibitor plus dopamine agonist combination class. See all MAO-B inhibitor plus dopamine agonist combination drugs at /class/mao-b-inhibitor-plus-dopamine-agonist-combination.

What development phase is Rasagiline mesylate plus Mirapex in?

Rasagiline mesylate plus Mirapex is FDA-approved (marketed).

What are the side effects of Rasagiline mesylate plus Mirapex?

Common side effects of Rasagiline mesylate plus Mirapex include Dyskinesia, Dizziness, Nausea, Hallucinations, Somnolence, Orthostatic hypotension.

What does Rasagiline mesylate plus Mirapex target?

Rasagiline mesylate plus Mirapex targets Monoamine oxidase B and dopamine D2/D3 receptors and is a MAO-B inhibitor plus dopamine agonist combination.

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