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R2: Lenalidomide + ixazomib maintenance

University of Leeds · Phase 3 active Small molecule

Lenalidomide and ixazomib work together as immunomodulatory and proteasome inhibitor agents to enhance anti-myeloma immune responses and suppress tumor cell proliferation in multiple myeloma maintenance therapy.

Lenalidomide and ixazomib work together as immunomodulatory and proteasome inhibitor agents to enhance anti-myeloma immune responses and suppress tumor cell proliferation in multiple myeloma maintenance therapy. Used for Multiple myeloma maintenance therapy (post-induction treatment).

At a glance

Generic nameR2: Lenalidomide + ixazomib maintenance
Also known asRevlimid, Ninlaro
SponsorUniversity of Leeds
Drug classImmunomodulatory agent + proteasome inhibitor combination
TargetCereblon (lenalidomide); 20S proteasome (ixazomib)
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

Lenalidomide is an immunomodulatory drug (IMiD) that enhances T-cell proliferation, NK cell activation, and TNF-α production while inhibiting angiogenesis. Ixazomib is a proteasome inhibitor that blocks NF-κB signaling and induces apoptosis in myeloma cells. Together in maintenance therapy, they provide dual mechanisms to prevent relapse and prolong progression-free survival in multiple myeloma patients.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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