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Placebo to DOR
DOR is a delta opioid receptor agonist that activates delta opioid receptors to modulate pain signaling and potentially provide analgesic effects.
DOR is a delta opioid receptor agonist that activates delta opioid receptors to modulate pain signaling and potentially provide analgesic effects. Used for Chronic pain (investigational).
At a glance
| Generic name | Placebo to DOR |
|---|---|
| Sponsor | Merck Sharp & Dohme LLC |
| Drug class | Delta opioid receptor agonist |
| Target | DOR (Delta opioid receptor) |
| Modality | Small molecule |
| Therapeutic area | Pain Management |
| Phase | Phase 3 |
Mechanism of action
Delta opioid receptors (DOR) are G-protein coupled receptors involved in pain modulation, mood regulation, and neuroprotection. Agonism at these receptors can produce analgesia through spinal and supraspinal mechanisms while potentially offering a different safety and abuse liability profile compared to mu opioid receptor agonists. This mechanism may provide pain relief with reduced respiratory depression and addiction potential.
Approved indications
- Chronic pain (investigational)
Common side effects
- Nausea
- Dizziness
- Headache
- Somnolence
Key clinical trials
- Switch to Doravirine/Islatravir (DOR/ISL) in Human Immunodeficiency Virus 1 (HIV-1) Participants Treated With Bictegravir/Emtricitabine/Tenofovir Alafenamide (BIC/FTC/TAF) (MK-8591A-018) (PHASE3)
- Study of Doravirine/Islatravir (DOR/ISL 100 mg/0.75 mg) to Evaluate the Antiretroviral Activity, Safety, and Tolerability in Treatment-Naïve Participants With Human Immunodeficiency Virus Type 1 (HIV-1) Infection (MK-8591A-020) (PHASE3)
- Clinical Evaluation of Integrated Chinese-Western Medicine for Infertility With DOR Patients in Women Achieving Natural Pregnancy (PHASE3)
- A Switch to Doravirine/Islatravir (DOR/ISL) in Participants With Human Immunodeficiency Virus Type 1 (HIV-1) Who Are Virologically Suppressed on Bictegravir/Emtricitabine/Tenofovir Alafenamide (BIC/FTC/TAF) (MK-8591A-052) (PHASE3)
- DOR/ISL in HIV-1 Antiretroviral Treatment-naïve Participants (MK-8591A-053) (PHASE3)
- The Clinical Trial of Electro-thumbtack Needle on Live Birth Rate in Patients With Ovarian Reserve Dysfunction (DOR) (NA)
- The Effect of VitC on IVF Outcome of DOR Patients (NA)
- Doravirine/Islatravir (DOR/ISL) in Heavily Treatment-Experienced (HTE) Participants for Human Immunodeficiency Virus Type 1 (HIV-1) Infection (MK-8591A-019) (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Placebo to DOR CI brief — competitive landscape report
- Placebo to DOR updates RSS · CI watch RSS
- Merck Sharp & Dohme LLC portfolio CI