Last reviewed · How we verify

pentolonium

unknown active ✓ Verified May 2026

pentolonium is a drug. It is currently in unknown development.

Pentolinium is a small molecule that acts as a nicotinic acetylcholine receptor antagonist. It is used as an antihypertensive drug, particularly during surgery or to control hypertensive crises.

At a glance

Generic namepentolonium
TargetNeuronal acetylcholine receptor subunit alpha-10, Neuronal acetylcholine receptor; alpha3/beta4
Therapeutic areaNeuroscience
Phaseunknown

Approved indications

No approved indications tracked.

Common side effects

No common side effects on file.

Competitive intelligence

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Frequently asked questions about pentolonium

What is pentolonium?

pentolonium is a pharmaceutical drug.

What development phase is pentolonium in?

pentolonium is in unknown.

What does pentolonium target?

pentolonium targets Neuronal acetylcholine receptor subunit alpha-10, Neuronal acetylcholine receptor; alpha3/beta4.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing