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PEG Asparaginase at two weeks interval

Rigshospitalet, Denmark · Phase 3 active Small molecule

PEG Asparaginase depletes the amino acid asparagine in the bloodstream, starving leukemic cells that cannot synthesize their own asparagine.

PEG Asparaginase depletes the amino acid asparagine in the bloodstream, starving leukemic cells that cannot synthesize their own asparagine. Used for Acute lymphoblastic leukemia (ALL), as part of combination chemotherapy.

At a glance

Generic namePEG Asparaginase at two weeks interval
Also known asOncaspar (PEG-Asparaginase)
SponsorRigshospitalet, Denmark
Drug classEnzyme (asparaginase)
TargetAsparagine
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

Asparaginase is an enzyme that catalyzes the hydrolysis of asparagine to aspartic acid and ammonia. Leukemic blasts, particularly in acute lymphoblastic leukemia (ALL), are dependent on exogenous asparagine for protein synthesis and cannot produce sufficient amounts endogenously. By depleting circulating asparagine, the drug selectively inhibits protein synthesis in leukemic cells while sparing normal cells that can synthesize asparagine. PEGylation extends the drug's half-life and reduces immunogenicity compared to native asparaginase.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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