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Parecoxib and remifentanil
Parecoxib and remifentanil is a COX-2 selective inhibitor (parecoxib) and opioid agonist (remifentanil) Small molecule drug developed by Ullevaal University Hospital. It is currently FDA-approved for Perioperative pain management and analgesia, Postoperative pain relief. Also known as: Dynastat.
Parecoxib is a selective COX-2 inhibitor that reduces pain and inflammation, while remifentanil is a potent opioid agonist that provides rapid analgesia and sedation.
Parecoxib is a selective COX-2 inhibitor that reduces pain and inflammation, while remifentanil is a potent opioid agonist that provides rapid analgesia and sedation. Used for Perioperative pain management, Postoperative analgesia.
At a glance
| Generic name | Parecoxib and remifentanil |
|---|---|
| Also known as | Dynastat |
| Sponsor | Ullevaal University Hospital |
| Drug class | COX-2 selective inhibitor (parecoxib) and opioid agonist (remifentanil) |
| Target | COX-2 (parecoxib); mu-opioid receptor (remifentanil) |
| Modality | Small molecule |
| Therapeutic area | Pain Management / Anesthesia |
| Phase | FDA-approved |
Mechanism of action
Parecoxib selectively inhibits cyclooxygenase-2 (COX-2), reducing prostaglandin synthesis and thereby decreasing pain and inflammation without affecting platelet function. Remifentanil is a synthetic opioid that binds to mu-opioid receptors in the central nervous system, providing rapid onset and offset analgesia and sedation due to its ester metabolism. Together, they provide multimodal analgesia for perioperative pain management.
Approved indications
- Perioperative pain management and analgesia
- Postoperative pain relief
Common side effects
- Nausea
- Vomiting
- Hypotension
- Respiratory depression
- Dizziness
- Headache
Key clinical trials
- Opioid-Free vs Opioid-Based Anesthesia in Bariatric Surgery (NA)
- Intravenous Dexamethasone and Dexmedetomidine on the Analgesic Efficacy of Erector Spinae Plane Block (NA)
- The Epigenetic Modification in OPRM1 on Postoperative Analgesia and Side Effect Induced by Sufentanil (PHASE4)
- Modulation of Remifentanil-induced Postinfusion Hyperalgesia (PHASE4)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Parecoxib and remifentanil CI brief — competitive landscape report
- Parecoxib and remifentanil updates RSS · CI watch RSS
- Ullevaal University Hospital portfolio CI
Frequently asked questions about Parecoxib and remifentanil
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Related
- Drug class: All COX-2 selective inhibitor (parecoxib) and opioid agonist (remifentanil) drugs
- Target: All drugs targeting COX-2 (parecoxib); mu-opioid receptor (remifentanil)
- Manufacturer: Ullevaal University Hospital — full pipeline
- Therapeutic area: All drugs in Pain Management / Anesthesia
- Indication: Drugs for Perioperative pain management and analgesia
- Indication: Drugs for Postoperative pain relief
- Also known as: Dynastat