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Ozempic® — mechanism of action

Hangzhou Zhongmei Huadong Pharmaceutical Co., Ltd.

Ozempic activates GLP-1 receptors to increase insulin secretion, slow gastric emptying, and reduce appetite, thereby lowering blood glucose levels in type 2 diabetes.

How ozempic works

Ozempic activates GLP-1 receptors to increase insulin secretion, slow gastric emptying, and reduce appetite, thereby lowering blood glucose levels in type 2 diabetes.

Detailed mechanism

Ozempic (semaglutide) is a GLP-1 receptor agonist that mimics glucagon-like peptide-1, a hormone that regulates blood sugar. It stimulates pancreatic beta cells to release insulin in response to elevated glucose, delays stomach emptying to reduce postprandial glucose spikes, and acts on the brain to suppress appetite and food intake. These combined effects improve glycemic control and promote weight loss.

Molecular targetGLP-1R (glucagon-like peptide-1 receptor)
Drug classGLP-1 receptor agonist
ModalitySmall molecule

See also

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing