Last reviewed · How we verify

Olumacostat Glasaretil Gel, 5.0%

Dermira, Inc. · Phase 3 active Small molecule

Olumacostat Glasaretil Gel, 5.0% is a SOAT1 inhibitor Small molecule drug developed by Dermira, Inc.. It is currently in Phase 3 development for Acne vulgaris. Also known as: DRM01, DRM01B.

Olumacostat glasaretil inhibits sebum production by blocking sterol O-acyltransferase (SOAT1), reducing lipid accumulation in sebaceous glands.

Olumacostat glasaretil inhibits sebum production by blocking sterol O-acyltransferase (SOAT1), reducing lipid accumulation in sebaceous glands. Used for Acne vulgaris.

At a glance

Generic nameOlumacostat Glasaretil Gel, 5.0%
Also known asDRM01, DRM01B
SponsorDermira, Inc.
Drug classSOAT1 inhibitor
TargetSOAT1 (sterol O-acyltransferase 1)
ModalitySmall molecule
Therapeutic areaDermatology
PhasePhase 3

Mechanism of action

The drug is a topical SOAT1 inhibitor that decreases sebaceous gland lipid synthesis and sebum secretion. By reducing sebum production, it addresses the underlying pathophysiology of acne and other sebum-related skin conditions. This mechanism targets a key driver of acne pathogenesis without systemic absorption.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:

Frequently asked questions about Olumacostat Glasaretil Gel, 5.0%

What is Olumacostat Glasaretil Gel, 5.0%?

Olumacostat Glasaretil Gel, 5.0% is a SOAT1 inhibitor drug developed by Dermira, Inc., indicated for Acne vulgaris.

How does Olumacostat Glasaretil Gel, 5.0% work?

Olumacostat glasaretil inhibits sebum production by blocking sterol O-acyltransferase (SOAT1), reducing lipid accumulation in sebaceous glands.

What is Olumacostat Glasaretil Gel, 5.0% used for?

Olumacostat Glasaretil Gel, 5.0% is indicated for Acne vulgaris.

Who makes Olumacostat Glasaretil Gel, 5.0%?

Olumacostat Glasaretil Gel, 5.0% is developed by Dermira, Inc. (see full Dermira, Inc. pipeline at /company/dermira-inc).

Is Olumacostat Glasaretil Gel, 5.0% also known as anything else?

Olumacostat Glasaretil Gel, 5.0% is also known as DRM01, DRM01B.

What drug class is Olumacostat Glasaretil Gel, 5.0% in?

Olumacostat Glasaretil Gel, 5.0% belongs to the SOAT1 inhibitor class. See all SOAT1 inhibitor drugs at /class/soat1-inhibitor.

What development phase is Olumacostat Glasaretil Gel, 5.0% in?

Olumacostat Glasaretil Gel, 5.0% is in Phase 3.

What are the side effects of Olumacostat Glasaretil Gel, 5.0%?

Common side effects of Olumacostat Glasaretil Gel, 5.0% include Application site irritation, Erythema, Dryness.

What does Olumacostat Glasaretil Gel, 5.0% target?

Olumacostat Glasaretil Gel, 5.0% targets SOAT1 (sterol O-acyltransferase 1) and is a SOAT1 inhibitor.

Related