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Non-selective NSAIDS
Non-selective NSAIDs inhibit both COX-1 and COX-2 enzymes to reduce prostaglandin synthesis, thereby decreasing inflammation, pain, and fever.
Non-selective NSAIDs inhibit both COX-1 and COX-2 enzymes to reduce prostaglandin synthesis, thereby decreasing inflammation, pain, and fever. Used for Mild to moderate pain, Rheumatoid arthritis, Osteoarthritis.
At a glance
| Generic name | Non-selective NSAIDS |
|---|---|
| Sponsor | Pfizer's Upjohn has merged with Mylan to form Viatris Inc. |
| Drug class | Non-selective NSAID |
| Target | COX-1 and COX-2 |
| Modality | Small molecule |
| Therapeutic area | Pain Management, Rheumatology, Cardiovascular |
| Phase | FDA-approved |
Mechanism of action
Non-selective NSAIDs block cyclooxygenase (COX) enzymes, which are responsible for producing prostaglandins—key mediators of inflammation, pain, and fever. By inhibiting both COX-1 and COX-2 isoforms, these drugs reduce prostaglandin levels systemically. This broad inhibition provides analgesic and anti-inflammatory effects but also increases the risk of gastrointestinal and cardiovascular adverse events compared to selective COX-2 inhibitors.
Approved indications
- Mild to moderate pain
- Rheumatoid arthritis
- Osteoarthritis
- Fever
- Dysmenorrhea
- Acute musculoskeletal pain
Common side effects
- Gastrointestinal bleeding or ulceration
- Dyspepsia
- Nausea
- Increased cardiovascular events (MI, stroke)
- Renal impairment
- Hypertension
- Headache
- Dizziness
Key clinical trials
- Multimodal Imaging and Biospecimen Collection for Low Back Pain (LBPB)
- Neuroregulators for the Treatment of Diseases Associated With Esophageal-brain-gut Axis Communication Abnormalities. (NA)
- Efficacy of NSAID vs. Steroid-NSAID Combo Post-Selective Laser Trabeculoplasty: Phase 4, Single-Center RCT (PHASE4)
- Adjunctive Celecoxib in Childhood-onset OCD Study (PHASE2)
- Post-authorization Safety Study of Etoricoxib and Other Anti-inflammatory Therapies in European Patients With Ankylosing Spondylitis (MK-0663-163)
- Milgamma® and Milgamma® Compositum Step-therapy in Patients With Acute Non-specific Low Back Pain Receiving Modern NSAID
- GI-Reasons- A Trial Of GI Safety Of Celecoxib Compared With Non-Selective Nonsteroidal Antiinflammatory Drugs (NSAIDS) (PHASE4)
- Open Label Comparative Study On Celecoxib Efficacy And Safety Vs Non-Selective NSAID In Acute Pain Due To Ankle Sprain (PHASE4)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Non-selective NSAIDS CI brief — competitive landscape report
- Non-selective NSAIDS updates RSS · CI watch RSS
- Pfizer's Upjohn has merged with Mylan to form Viatris Inc. portfolio CI