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mTOR inhibitor (everolimus)
mTOR inhibitor (everolimus) is a mTOR inhibitor Small molecule drug developed by Hannover Medical School. It is currently FDA-approved for Advanced renal cell carcinoma, Breast cancer (hormone receptor-positive, HER2-negative), Neuroendocrine tumors of pancreatic origin. Also known as: switch immunosuppression to everolimus.
Everolimus inhibits mTOR (mammalian target of rapamycin), a key protein kinase that regulates cell growth and proliferation.
Everolimus inhibits mTOR (mammalian target of rapamycin), a key protein kinase that regulates cell growth and proliferation. Used for Advanced renal cell carcinoma, Breast cancer (hormone receptor-positive, HER2-negative), Neuroendocrine tumors of pancreatic origin.
At a glance
| Generic name | mTOR inhibitor (everolimus) |
|---|---|
| Also known as | switch immunosuppression to everolimus |
| Sponsor | Hannover Medical School |
| Drug class | mTOR inhibitor |
| Target | mTOR (mammalian target of rapamycin) |
| Modality | Small molecule |
| Therapeutic area | Oncology |
| Phase | FDA-approved |
Mechanism of action
mTOR is a central regulator of cell metabolism, growth, and survival. By blocking mTOR signaling, everolimus suppresses cell proliferation and angiogenesis, making it effective in cancers and certain proliferative diseases. It also has immunomodulatory effects that enhance T-cell activation in some contexts.
Approved indications
- Advanced renal cell carcinoma
- Breast cancer (hormone receptor-positive, HER2-negative)
- Neuroendocrine tumors of pancreatic origin
- Subependymal giant cell astrocytoma (SEGA) associated with tuberous sclerosis complex
- Renal angiomyolipoma associated with tuberous sclerosis complex
Common side effects
- Stomatitis/mouth ulcers
- Rash
- Diarrhea
- Fatigue
- Nausea
- Anemia
- Hyperglycemia
- Hyperlipidemia
- Infections
Key clinical trials
- Testing Lutetium Lu 177 Dotatate in Patients With Somatostatin Receptor Positive Advanced Bronchial Neuroendocrine Tumors (PHASE2)
- Comparing Retreatment of 177Lu-DOTATATE PRRT Versus the Usual Treatment in Patients With Metastatic Unresectable Gastroenteropancreatic Neuroendocrine Tumors, NET RETREAT Trial (PHASE2)
- A Study to Evaluate Axatilimab Versus Best Available Therapy in Participants With Chronic Graft Versus Host Disease After at Least 2 Prior Lines of Systemic Therapy (PHASE3)
- A Study to Evaluate Axatilimab Versus Best Available Therapy in Pediatric Participants With Chronic Graft-Versus-Host Disease After at Least 2 Prior Lines of Systemic Therapy (AGAVE-256) (PHASE2)
- Phase 1/2 Study to Evaluate EP0062 as Monotherapy and in Combination in Patients With Advanced or Metastatic AR+/HER-2-/ER+ Breast Cancer (PHASE1, PHASE2)
- Lenvatinib and Everolimus in Treating Patients With Advanced, Unresectable Carcinoid Tumors (PHASE2)
- Trametinib and Everolimus for Treatment of Pediatric and Young Adult Patients With Recurrent Gliomas (PNOC021) (PHASE1)
- Lenvatinib With Everolimus Versus Cabozantinib for Second-Line or Third-Line Treatment of Metastatic Renal Cell Cancer (PHASE2)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- mTOR inhibitor (everolimus) CI brief — competitive landscape report
- mTOR inhibitor (everolimus) updates RSS · CI watch RSS
- Hannover Medical School portfolio CI
Frequently asked questions about mTOR inhibitor (everolimus)
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Related
- Drug class: All mTOR inhibitor drugs
- Target: All drugs targeting mTOR (mammalian target of rapamycin)
- Manufacturer: Hannover Medical School — full pipeline
- Therapeutic area: All drugs in Oncology
- Indication: Drugs for Advanced renal cell carcinoma
- Indication: Drugs for Breast cancer (hormone receptor-positive, HER2-negative)
- Indication: Drugs for Neuroendocrine tumors of pancreatic origin
- Also known as: switch immunosuppression to everolimus
- Compare: mTOR inhibitor (everolimus) vs similar drugs
- Pricing: mTOR inhibitor (everolimus) cost, discount & access