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midazolam + pethidine

Erasme University Hospital · FDA-approved active Small molecule

Midazolam and pethidine together provide sedation and analgesia by acting as a benzodiazepine and opioid, respectively, enhancing CNS depression for procedural or acute pain management.

Midazolam and pethidine together provide sedation and analgesia by acting as a benzodiazepine and opioid, respectively, enhancing CNS depression for procedural or acute pain management. Used for Procedural sedation and analgesia, Acute pain management with sedation.

At a glance

Generic namemidazolam + pethidine
SponsorErasme University Hospital
Drug classBenzodiazepine + Opioid combination
TargetGABA-A receptor (midazolam); mu opioid receptor (pethidine)
ModalitySmall molecule
Therapeutic areaAnesthesia/Sedation, Pain Management
PhaseFDA-approved

Mechanism of action

Midazolam is a short-acting benzodiazepine that potentiates GABA-A receptor signaling to produce sedation, anxiolysis, and amnesia. Pethidine (meperidine) is a synthetic opioid that binds mu opioid receptors to produce analgesia and additional sedation. The combination is used clinically to achieve balanced sedation and pain relief, particularly in procedural settings.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results