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mFOLFIRINOX regimen

Revolution Medicines, Inc. · Phase 3 active Small molecule

mFOLFIRINOX is a chemotherapy regimen combining 5-fluorouracil, leucovorin, irinotecan, and oxaliplatin to inhibit DNA synthesis and induce apoptosis in cancer cells.

mFOLFIRINOX is a chemotherapy regimen combining 5-fluorouracil, leucovorin, irinotecan, and oxaliplatin to inhibit DNA synthesis and induce apoptosis in cancer cells. Used for Metastatic pancreatic cancer, Metastatic colorectal cancer, Gastric cancer.

At a glance

Generic namemFOLFIRINOX regimen
Also known asmodified FOLFIRINOX regimen, modified regimen of oxaliplatin, leucovorin, irinotecan, and fluorouracil (5-FU), Folic acid, 5- fluorouracil, irinotecan and oxaliplatin, Oxaliplatin, Irinotecan
SponsorRevolution Medicines, Inc.
Drug classCombination chemotherapy regimen
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

This is a combination chemotherapy regimen where each agent targets cancer cell proliferation through different mechanisms: 5-FU and leucovorin inhibit thymidylate synthase, irinotecan inhibits topoisomerase I, and oxaliplatin causes DNA cross-linking. The 'modified' (mFOLFIRINOX) version typically refers to adjusted dosing schedules designed to improve tolerability while maintaining efficacy compared to the standard regimen.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results