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Metformin, glyburide and insulin
Metformin, glyburide and insulin is a Antidiabetic combination therapy (biguanide + sulfonylurea + insulin) Small molecule drug developed by Université de Sherbrooke. It is currently in Phase 3 development for Type 2 diabetes mellitus.
This combination therapy addresses type 2 diabetes through three complementary mechanisms: metformin reduces hepatic glucose production, glyburide stimulates pancreatic insulin secretion, and insulin provides direct glucose-lowering action.
This combination therapy addresses type 2 diabetes through three complementary mechanisms: metformin reduces hepatic glucose production, glyburide stimulates pancreatic insulin secretion, and insulin provides direct glucose-lowering action. Used for Type 2 diabetes mellitus.
At a glance
| Generic name | Metformin, glyburide and insulin |
|---|---|
| Sponsor | Université de Sherbrooke |
| Drug class | Antidiabetic combination therapy (biguanide + sulfonylurea + insulin) |
| Modality | Small molecule |
| Therapeutic area | Diabetes |
| Phase | Phase 3 |
Mechanism of action
Metformin is a biguanide that decreases hepatic gluconeogenesis and improves insulin sensitivity. Glyburide is a sulfonylurea that stimulates beta cells to release endogenous insulin. Insulin provides exogenous glucose control. Together, these agents target multiple pathways in diabetes pathophysiology—hepatic glucose output, endogenous insulin secretion, and peripheral glucose uptake.
Approved indications
- Type 2 diabetes mellitus
Common side effects
- Hypoglycemia
- Gastrointestinal disturbance (metformin)
- Weight gain (insulin, glyburide)
- Lactic acidosis (metformin, rare)
Key clinical trials
- Comparative Effectiveness and Safety of Four Second Line Pharmacological Strategies in Type 2 Diabetes Study
- Metabolic Analysis for Treatment Choice in Gestational Diabetes Mellitus (PHASE4)
- Durability of Combination Therapy With Exenatide/Pioglitazone/Metformin vs. Conventional Therapy in New Onset T2DM (PHASE4)
- BESTMED: Observational Evaluation of Second Line Therapy Medications in Diabetes
- Gestational Diabetes: Insulin or Oral Hypoglycemic Agents? (PHASE3)
- Preservation of Beta-cell Function in Type 2 Diabetes Mellitus (NA)
- An Observational Study of Type II Diabetics Treated With Dual Therapy With or Without Sitagliptin (Januvia®/Xelevia®, MK-0431-201)
- Efficacy and Safety of Lixisenatide Versus Placebo on Top of Basal Insulin and/or Oral Antidiabetic Treatment in Older Type 2 Diabetic Patients (PHASE3)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Metformin, glyburide and insulin CI brief — competitive landscape report
- Metformin, glyburide and insulin updates RSS · CI watch RSS
- Université de Sherbrooke portfolio CI
Frequently asked questions about Metformin, glyburide and insulin
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Related
- Drug class: All Antidiabetic combination therapy (biguanide + sulfonylurea + insulin) drugs
- Manufacturer: Université de Sherbrooke — full pipeline
- Therapeutic area: All drugs in Diabetes
- Indication: Drugs for Type 2 diabetes mellitus
- Compare: Metformin, glyburide and insulin vs similar drugs
- Pricing: Metformin, glyburide and insulin cost, discount & access