Last reviewed · How we verify

Melanex (METAHEXAMIDE)

Phase 2 active Small molecule

Melanex (generic name: METAHEXAMIDE) is a metahexamide drug. It is currently in Phase 2 development for Chloasma, Discoloration of skin.

Melanex works by inhibiting the enzyme tyrosinase, which is involved in the production of melanin, the pigment responsible for skin color.

Melanex, also known as metahexamide, is a small molecule drug in the metahexamide class. It is used to treat Chloasma and skin discoloration. The commercial status of Melanex is currently unknown, and it is not clear if it is patented or available as a generic. Further information on its approval status, half-life, and bioavailability is also not available. As a result, key safety considerations and pharmacological details are not well established.

Likelihood of approval
15.3% vs 15.3% industry baseline
If approved by FDA: likely 2031–2034
Steps remaining: Phase 3 → NDA/BLA submission
Confidence: Medium
Why this estimate
  • Baseline phase 2 → approval rate +15.3pp
    Industry-wide phase 2 drugs reach approval ~15.3% of the time (BIO/Informa 2023 industry benchmark across all therapeutic areas).
Predicted approval windows by jurisdiction (conditional on FDA approval)
Regulator Country Likely year Lag vs FDA
FDA US 2031–2034
EMA EU 2032–2035 +0.7 yr
MHRA GB 2032–2035 +0.7 yr
Health Canada CA 2032–2036 +0.9 yr
TGA AU 2032–2036 +1.2 yr
PMDA JP 2032–2036 +1.5 yr
NMPA CN 2033–2037 +2.3 yr
MFDS KR 2032–2036 +1.4 yr
CDSCO IN 2032–2037 +1.8 yr
ANVISA BR 2033–2037 +2.3 yr

Hover any row for the lag rationale. Lag estimates are reduced when the drug has FDA Breakthrough or EMA PRIME designation (sponsors file globally in parallel).

Estimate based on the BIO/Informa industry phase transition rates plus per-drug modifiers for therapeutic area, sponsor type, FDA designations, mechanism, and trial design. Per-jurisdiction lags from Tufts CSDD international approval studies. Not investment, clinical or regulatory advice. Methodology: /methodology#likelihood.

At a glance

Generic nameMETAHEXAMIDE
Drug classmetahexamide
ModalitySmall molecule
Therapeutic areaDermatology
PhasePhase 2

Mechanism of action

Think of melanin like the paint that colors your skin. Tyrosinase is the brush that helps spread the paint. Melanex blocks the brush, so less paint is applied, resulting in lighter skin color. This can help reduce the appearance of Chloasma and skin discoloration.

Approved indications

Common side effects

No common side effects on file.

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

Competitive intelligence

For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:

Frequently asked questions about Melanex

What is Melanex?

Melanex (METAHEXAMIDE) is a metahexamide drug, indicated for Chloasma, Discoloration of skin.

How does Melanex work?

Melanex works by inhibiting the enzyme tyrosinase, which is involved in the production of melanin, the pigment responsible for skin color.

What is Melanex used for?

Melanex is indicated for Chloasma, Discoloration of skin.

What is the generic name of Melanex?

METAHEXAMIDE is the generic (nonproprietary) name of Melanex.

What drug class is Melanex in?

Melanex belongs to the metahexamide class. See all metahexamide drugs at /class/metahexamide.

What development phase is Melanex in?

Melanex is in Phase 2.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing