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Mesalazine(asacol 800 mg)
Mesalazine(asacol 800 mg) is a 5-aminosalicylic acid (5-ASA) agent Small molecule drug developed by Tehran University of Medical Sciences. It is currently FDA-approved for Ulcerative colitis, mild to moderate, Crohn's disease, mild to moderate, Maintenance of remission in inflammatory bowel disease.
Mesalazine reduces intestinal inflammation by inhibiting prostaglandin and leukotriene production in the colon.
Mesalazine reduces intestinal inflammation by inhibiting prostaglandin and leukotriene production in the colon. Used for Ulcerative colitis (induction and maintenance of remission), Crohn's disease (colonic involvement).
At a glance
| Generic name | Mesalazine(asacol 800 mg) |
|---|---|
| Sponsor | Tehran University of Medical Sciences |
| Drug class | 5-aminosalicylic acid (5-ASA) agent |
| Target | Prostaglandin and leukotriene synthesis; nuclear factor-kappa B (NF-κB) pathway |
| Modality | Small molecule |
| Therapeutic area | Gastroenterology |
| Phase | FDA-approved |
Mechanism of action
Mesalazine (5-aminosalicylic acid) is a topical anti-inflammatory agent that acts locally in the colon to suppress inflammatory mediators and reduce immune cell activation. It inhibits nuclear factor-kappa B (NF-κB) signaling and decreases production of pro-inflammatory cytokines, thereby reducing mucosal inflammation in inflammatory bowel disease.
Approved indications
- Ulcerative colitis, mild to moderate
- Crohn's disease, mild to moderate
- Maintenance of remission in inflammatory bowel disease
Common side effects
- Headache
- Abdominal pain
- Diarrhea
- Nausea
- Rash
- Nephrotoxicity (rare)
Key clinical trials
- Adherence of a 1.600 mg Single Tablet 5-ASA Treatment of Ulcerative Colitis (PHASE4)
- Sulfamethoxazole Drug Interaction Study With MMX® Mesalazine/Mesalamine (PHASE1)
- Efficacy and Safety of SPD476 in Maintaining Remission in Patients With Ulcerative Colitis (PHASE3)
- The Colitis Once Daily Asacol Study (PHASE3)
- Cimzia Versus Mesalamine for Crohn's Recurrence (PHASE4)
- Efficacy and Safety of Asacol™ 4.8 g/Day (800 mg Tablets) for the Treatment of Active Ulcerative Colitis (PHASE3)
- Chemopreventive Action of Mesalazine on Colorectal Cancer: a Pilot Study for an "in Vivo" Evaluation of the Molecular Effects on β-catenin Signaling Pathway. (PHASE2)
- Effects of Mesalamine and Amitriptyline on Irritable Bowel Syndrome (PHASE4)
Primary sources
Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.
| Source | Used for |
|---|---|
| ClinicalTrials.gov | Trial enrolment, design, endpoints, results |
Competitive intelligence
For the full competitive landscape — auto-detected comparators, recent regulatory actions across the set, upcoming PDUFA, patent timeline, sponsor landscape:
- Mesalazine(asacol 800 mg) CI brief — competitive landscape report
- Mesalazine(asacol 800 mg) updates RSS · CI watch RSS
- Tehran University of Medical Sciences portfolio CI
Frequently asked questions about Mesalazine(asacol 800 mg)
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Related
- Drug class: All 5-aminosalicylic acid (5-ASA) agent drugs
- Target: All drugs targeting Prostaglandin and leukotriene synthesis; nuclear factor-kappa B (NF-κB) pathway
- Manufacturer: Tehran University of Medical Sciences — full pipeline
- Therapeutic area: All drugs in Gastroenterology
- Indication: Drugs for Ulcerative colitis, mild to moderate
- Indication: Drugs for Crohn's disease, mild to moderate
- Indication: Drugs for Maintenance of remission in inflammatory bowel disease
- Compare: Mesalazine(asacol 800 mg) vs similar drugs
- Pricing: Mesalazine(asacol 800 mg) cost, discount & access