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Levosimendan infusion

AHEPA University Hospital · FDA-approved active Small molecule

Levosimendan infusion is a Calcium sensitizer / inodilator Small molecule drug developed by AHEPA University Hospital. It is currently FDA-approved for Acute decompensated heart failure, Cardiogenic shock.

Levosimendan is a calcium sensitizer that increases the force of cardiac muscle contraction without increasing oxygen consumption, while also causing vasodilation through opening of ATP-sensitive potassium channels.

Levosimendan is a calcium sensitizer that increases the force of cardiac muscle contraction without increasing oxygen consumption, while also causing vasodilation through opening of ATP-sensitive potassium channels. Used for Acute decompensated heart failure.

At a glance

Generic nameLevosimendan infusion
SponsorAHEPA University Hospital
Drug classCalcium sensitizer / inodilator
TargetCardiac troponin C; ATP-sensitive potassium channels
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Levosimendan binds to cardiac troponin C and enhances the interaction between actin and myosin filaments, thereby increasing myocardial contractility. Simultaneously, it opens ATP-sensitive potassium channels in vascular smooth muscle, producing vasodilation and reducing cardiac afterload. This dual mechanism improves cardiac output while reducing myocardial oxygen demand.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Levosimendan infusion

What is Levosimendan infusion?

Levosimendan infusion is a Calcium sensitizer / inodilator drug developed by AHEPA University Hospital, indicated for Acute decompensated heart failure, Cardiogenic shock.

How does Levosimendan infusion work?

Levosimendan is a calcium sensitizer that increases the force of cardiac muscle contraction without increasing oxygen consumption, while also causing vasodilation through opening of ATP-sensitive potassium channels.

What is Levosimendan infusion used for?

Levosimendan infusion is indicated for Acute decompensated heart failure, Cardiogenic shock.

Who makes Levosimendan infusion?

Levosimendan infusion is developed and marketed by AHEPA University Hospital (see full AHEPA University Hospital pipeline at /company/ahepa-university-hospital).

What drug class is Levosimendan infusion in?

Levosimendan infusion belongs to the Calcium sensitizer / inodilator class. See all Calcium sensitizer / inodilator drugs at /class/calcium-sensitizer-inodilator.

What development phase is Levosimendan infusion in?

Levosimendan infusion is FDA-approved (marketed).

What are the side effects of Levosimendan infusion?

Common side effects of Levosimendan infusion include Headache, Hypotension, Arrhythmias, Nausea.

What does Levosimendan infusion target?

Levosimendan infusion targets Cardiac troponin C; ATP-sensitive potassium channels and is a Calcium sensitizer / inodilator.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing