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LCP-tacrolimus QD + MMF BID

University Hospital, Limoges · FDA-approved active Small molecule

LCP-tacrolimus is a prolonged-release formulation of tacrolimus combined with mycophenolate mofetil (MMF) to suppress T-cell mediated immune responses and prevent organ rejection.

LCP-tacrolimus is a prolonged-release formulation of tacrolimus combined with mycophenolate mofetil (MMF) to suppress T-cell mediated immune responses and prevent organ rejection. Used for Prevention of organ rejection in transplant recipients (kidney, heart, liver transplantation).

At a glance

Generic nameLCP-tacrolimus QD + MMF BID
SponsorUniversity Hospital, Limoges
Drug classCalcineurin inhibitor + antimetabolite combination
TargetCalcineurin (tacrolimus); IMPDH type II (mycophenolate mofetil)
ModalitySmall molecule
Therapeutic areaImmunology / Transplantation
PhaseFDA-approved

Mechanism of action

Tacrolimus is a calcineurin inhibitor that blocks T-cell activation by inhibiting IL-2 production, while MMF is an inosine monophosphate dehydrogenase inhibitor that selectively suppresses lymphocyte proliferation. The LCP (Lipid Conjugate Platform) formulation provides once-daily dosing of tacrolimus, improving adherence in immunosuppressive regimens. Together, these agents provide complementary immunosuppression for transplant rejection prevention.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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