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Latanoprost, Dorzolamide

Azienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia · FDA-approved active Small molecule

This combination reduces intraocular pressure by increasing uveoscleral outflow of aqueous humor (latanoprost) and decreasing aqueous humor production (dorzolamide).

This combination reduces intraocular pressure by increasing uveoscleral outflow of aqueous humor (latanoprost) and decreasing aqueous humor production (dorzolamide). Used for Open-angle glaucoma, Ocular hypertension.

At a glance

Generic nameLatanoprost, Dorzolamide
Also known as- Latanoprost, a prostaglandin analogue, - Dorzolamide, a potent inhibitor of carbonic anhydrase II
SponsorAzienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia
Drug classProstaglandin analog + Carbonic anhydrase inhibitor combination
TargetProstaglandin F receptor (FP receptor) and Carbonic anhydrase II
ModalitySmall molecule
Therapeutic areaOphthalmology
PhaseFDA-approved

Mechanism of action

Latanoprost is a prostaglandin F analog that binds to prostaglandin F receptors and enhances drainage of aqueous humor through the uveoscleral pathway. Dorzolamide is a carbonic anhydrase inhibitor that reduces aqueous humor secretion by inhibiting carbonic anhydrase in the ciliary body. Together, these complementary mechanisms provide additive intraocular pressure reduction.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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