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IV TXA

Massachusetts General Hospital · FDA-approved active Small molecule

IV TXA (tranexamic acid) inhibits fibrinolysis by blocking plasminogen activation, thereby reducing bleeding.

IV TXA (tranexamic acid) inhibits fibrinolysis by blocking plasminogen activation, thereby reducing bleeding. Used for Acute hemorrhage and trauma, Perioperative blood loss reduction, Heavy menstrual bleeding.

At a glance

Generic nameIV TXA
SponsorMassachusetts General Hospital
Drug classAntifibrinolytic agent
TargetPlasminogen / Plasmin
ModalitySmall molecule
Therapeutic areaHematology / Hemostasis
PhaseFDA-approved

Mechanism of action

Tranexamic acid is a competitive inhibitor of plasminogen and plasmin, which are enzymes responsible for breaking down fibrin clots. By preventing fibrin degradation, it stabilizes clots and reduces hemorrhage. It is commonly used intravenously in acute bleeding situations, trauma, and perioperative settings to minimize blood loss.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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