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Iron isomaltoside/ferric derisomaltose

Pharmacosmos A/S · Phase 3 active Small molecule

Iron isomaltoside/ferric derisomaltose is a Iron replacement therapy Small molecule drug developed by Pharmacosmos A/S. It is currently in Phase 3 development for Iron deficiency anemia in adult patients, Iron deficiency anemia in pediatric patients. Also known as: Monofer®, Monoferric®, Monover®, Monofar®, Monoferro®.

Iron isomaltoside delivers ferric iron complexed with isomaltoside, a carbohydrate polymer, to replenish iron stores and treat iron deficiency anemia.

Iron isomaltoside delivers ferric iron complexed with isomaltoside, a carbohydrate polymer, to replenish iron stores and treat iron deficiency anemia. Used for Iron deficiency anemia in adult patients, Iron deficiency anemia in pediatric patients.

At a glance

Generic nameIron isomaltoside/ferric derisomaltose
Also known asMonofer®, Monoferric®, Monover®, Monofar®, Monoferro®
SponsorPharmacosmos A/S
Drug classIron replacement therapy
TargetIron metabolism pathway; ferric iron (Fe3+)
ModalitySmall molecule
Therapeutic areaHematology
PhasePhase 3

Mechanism of action

The isomaltoside carbohydrate shell protects the ferric iron core during transit through the gastrointestinal tract and facilitates absorption and cellular uptake. Once absorbed, the iron is released and incorporated into hemoglobin and other iron-dependent proteins to restore oxygen-carrying capacity and correct anemia. This formulation allows for rapid iron repletion with improved tolerability compared to traditional iron salts.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Iron isomaltoside/ferric derisomaltose

What is Iron isomaltoside/ferric derisomaltose?

Iron isomaltoside/ferric derisomaltose is a Iron replacement therapy drug developed by Pharmacosmos A/S, indicated for Iron deficiency anemia in adult patients, Iron deficiency anemia in pediatric patients.

How does Iron isomaltoside/ferric derisomaltose work?

Iron isomaltoside delivers ferric iron complexed with isomaltoside, a carbohydrate polymer, to replenish iron stores and treat iron deficiency anemia.

What is Iron isomaltoside/ferric derisomaltose used for?

Iron isomaltoside/ferric derisomaltose is indicated for Iron deficiency anemia in adult patients, Iron deficiency anemia in pediatric patients.

Who makes Iron isomaltoside/ferric derisomaltose?

Iron isomaltoside/ferric derisomaltose is developed by Pharmacosmos A/S (see full Pharmacosmos A/S pipeline at /company/pharmacosmos-a-s).

Is Iron isomaltoside/ferric derisomaltose also known as anything else?

Iron isomaltoside/ferric derisomaltose is also known as Monofer®, Monoferric®, Monover®, Monofar®, Monoferro®.

What drug class is Iron isomaltoside/ferric derisomaltose in?

Iron isomaltoside/ferric derisomaltose belongs to the Iron replacement therapy class. See all Iron replacement therapy drugs at /class/iron-replacement-therapy.

What development phase is Iron isomaltoside/ferric derisomaltose in?

Iron isomaltoside/ferric derisomaltose is in Phase 3.

What are the side effects of Iron isomaltoside/ferric derisomaltose?

Common side effects of Iron isomaltoside/ferric derisomaltose include Nausea, Abdominal pain, Diarrhea, Headache, Injection site reactions (if parenteral formulation).

What does Iron isomaltoside/ferric derisomaltose target?

Iron isomaltoside/ferric derisomaltose targets Iron metabolism pathway; ferric iron (Fe3+) and is a Iron replacement therapy.

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