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Iron isomaltoside

Thomas Jefferson University · FDA-approved active Small molecule

Iron isomaltoside is an iron replacement therapy that delivers ferric iron complexed with isomaltoside, allowing efficient absorption and utilization for hemoglobin synthesis in iron-deficient patients.

Iron isomaltoside is an iron replacement therapy that delivers ferric iron complexed with isomaltoside, allowing efficient absorption and utilization for hemoglobin synthesis in iron-deficient patients. Used for Iron deficiency anemia in patients with chronic kidney disease, Iron deficiency anemia in patients intolerant to or non-responsive to oral iron.

At a glance

Generic nameIron isomaltoside
Also known asFerric derisomaltose, Monofer, Intravenous iron isomaltoside
SponsorThomas Jefferson University
Drug classIron replacement agent
TargetIron (Fe3+) / transferrin receptor
ModalitySmall molecule
Therapeutic areaHematology
PhaseFDA-approved

Mechanism of action

Iron isomaltoside is a carbohydrate-based iron complex that provides bioavailable iron for patients with iron deficiency. The isomaltoside carbohydrate shell protects the iron core during transit through the gastrointestinal tract and facilitates cellular uptake via transferrin-mediated pathways, enabling rapid repletion of iron stores and restoration of oxygen-carrying capacity.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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