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Infliximab (Remicade)

University of California, San Diego · FDA-approved active Small molecule

Infliximab is a monoclonal antibody that binds to and neutralizes tumor necrosis factor-alpha (TNF-α), a key inflammatory cytokine.

Infliximab is a monoclonal antibody that binds to and neutralizes tumor necrosis factor-alpha (TNF-α), a key inflammatory cytokine. Used for Rheumatoid arthritis, Crohn's disease, Ulcerative colitis.

At a glance

Generic nameInfliximab (Remicade)
Also known asRemicade, SCH 215596
SponsorUniversity of California, San Diego
Drug classTNF-α inhibitor (monoclonal antibody)
TargetTNF-α (Tumor Necrosis Factor-alpha)
ModalitySmall molecule
Therapeutic areaImmunology
PhaseFDA-approved

Mechanism of action

By blocking TNF-α, infliximab reduces the inflammatory cascade that drives autoimmune and inflammatory diseases. This TNF-α inhibition decreases immune cell activation, reduces production of other inflammatory mediators, and promotes apoptosis of inflammatory cells. The drug is effective in conditions where TNF-α plays a central pathogenic role, including rheumatoid arthritis, inflammatory bowel disease, and psoriasis.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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