Last reviewed · How we verify

Isindone (INDOPROFEN)

FDA-approved withdrawn Small molecule Quality 17/100

Indoprofen (Isindone) is a marketed drug that uniquely inhibits the pyruvate kinase PKM enzyme, setting it apart in the NSAID class. Its key strength lies in its distinct mechanism of action, which differentiates it from competitors such as ibuprofen, naproxen, ketoprofen, and fenoprofen, all of which are either off-patent or have significant generic competition. The primary risk is the key composition patent expiry in 2028, which could lead to increased competition from generics.

At a glance

Generic nameINDOPROFEN
Drug classindoprofen
TargetPyruvate kinase PKM, Fatty acid-binding protein, liver, Luciferin 4-monooxygenase
ModalitySmall molecule
Therapeutic areaGastroenterology
PhaseFDA-approved
First approval1979

Approved indications

No approved indications tracked.

Common side effects

No common side effects on file.

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
FDA labelMechanism, indications, dosing, boxed warnings, drug interactions

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