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Imiquimod 5%: manufactured by Apotex

Apotex Inc. · Phase 3 active Small molecule

Imiquimod 5%: manufactured by Apotex is a TLR7 agonist Small molecule drug developed by Apotex Inc.. It is currently in Phase 3 development for Actinic keratosis, Basal cell carcinoma (superficial and nodular), Genital warts (external).

Imiquimod is a toll-like receptor 7 (TLR7) agonist that activates innate immune responses to treat skin lesions and certain cancers.

Imiquimod is a toll-like receptor 7 (TLR7) agonist that activates innate immune responses to treat skin lesions and certain cancers. Used for Actinic keratosis, Basal cell carcinoma (superficial and nodular), Genital warts (external).

At a glance

Generic nameImiquimod 5%: manufactured by Apotex
SponsorApotex Inc.
Drug classTLR7 agonist
TargetTLR7 (Toll-like receptor 7)
ModalitySmall molecule
Therapeutic areaDermatology, Oncology, Immunology
PhasePhase 3

Mechanism of action

Imiquimod binds to TLR7 on immune cells, triggering the production of interferon-alpha and other cytokines that enhance local immune activation. This stimulates both innate and adaptive immune responses against abnormal cells or viral-infected cells in the skin. The resulting inflammation and immune cell infiltration lead to clearance of targeted lesions.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about Imiquimod 5%: manufactured by Apotex

What is Imiquimod 5%: manufactured by Apotex?

Imiquimod 5%: manufactured by Apotex is a TLR7 agonist drug developed by Apotex Inc., indicated for Actinic keratosis, Basal cell carcinoma (superficial and nodular), Genital warts (external).

How does Imiquimod 5%: manufactured by Apotex work?

Imiquimod is a toll-like receptor 7 (TLR7) agonist that activates innate immune responses to treat skin lesions and certain cancers.

What is Imiquimod 5%: manufactured by Apotex used for?

Imiquimod 5%: manufactured by Apotex is indicated for Actinic keratosis, Basal cell carcinoma (superficial and nodular), Genital warts (external), Cutaneous T-cell lymphoma (mycosis fungoides).

Who makes Imiquimod 5%: manufactured by Apotex?

Imiquimod 5%: manufactured by Apotex is developed by Apotex Inc. (see full Apotex Inc. pipeline at /company/apotex-inc).

What drug class is Imiquimod 5%: manufactured by Apotex in?

Imiquimod 5%: manufactured by Apotex belongs to the TLR7 agonist class. See all TLR7 agonist drugs at /class/tlr7-agonist.

What development phase is Imiquimod 5%: manufactured by Apotex in?

Imiquimod 5%: manufactured by Apotex is in Phase 3.

What are the side effects of Imiquimod 5%: manufactured by Apotex?

Common side effects of Imiquimod 5%: manufactured by Apotex include Local skin irritation (erythema, erosion, excoriation), Pruritus, Burning sensation, Scabbing/crusting, Systemic flu-like symptoms (fatigue, fever, myalgia), Lymphadenopathy.

What does Imiquimod 5%: manufactured by Apotex target?

Imiquimod 5%: manufactured by Apotex targets TLR7 (Toll-like receptor 7) and is a TLR7 agonist.

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