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hypoglycemic Agents(metformin)

First Affiliated Hospital of Wenzhou Medical University · FDA-approved active Small molecule ✓ Verified Jun 2026

hypoglycemic Agents(metformin) is a Biguanide Small molecule drug developed by First Affiliated Hospital of Wenzhou Medical University. It is currently FDA-approved for Type 2 diabetes mellitus, Prediabetes (off-label or prevention studies).

Metformin reduces hepatic glucose production and improves insulin sensitivity in peripheral tissues, thereby lowering blood glucose levels in type 2 diabetes.

Metformin is a small molecule hypoglycemic agent used to treat Type 2 Diabetes Mellitus, as indicated by its study in various clinical trials on ClinicalTrials.gov. Its mechanism of action is not specified in the provided facts, but it is classified as a small molecule according to ChEMBL.

At a glance

Generic namehypoglycemic Agents(metformin)
SponsorFirst Affiliated Hospital of Wenzhou Medical University
Drug classBiguanide
TargetAMP-activated protein kinase (AMPK); complex I of the mitochondrial electron transport chain
ModalitySmall molecule
Therapeutic areaEndocrinology / Diabetes
PhaseFDA-approved

Mechanism of action

Metformin is a biguanide that primarily works by decreasing gluconeogenesis in the liver and enhancing glucose uptake and utilization in muscle and adipose tissue. It does not stimulate insulin secretion, making it weight-neutral and useful in combination with other agents. The drug may also improve insulin sensitivity through activation of AMP-activated protein kinase (AMPK) and modulation of mitochondrial function.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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Frequently asked questions about hypoglycemic Agents(metformin)

What is hypoglycemic Agents(metformin)?

hypoglycemic Agents(metformin) is a Biguanide drug developed by First Affiliated Hospital of Wenzhou Medical University, indicated for Type 2 diabetes mellitus, Prediabetes (off-label or prevention studies).

How does hypoglycemic Agents(metformin) work?

Metformin reduces hepatic glucose production and improves insulin sensitivity in peripheral tissues, thereby lowering blood glucose levels in type 2 diabetes.

What is hypoglycemic Agents(metformin) used for?

hypoglycemic Agents(metformin) is indicated for Type 2 diabetes mellitus, Prediabetes (off-label or prevention studies).

Who makes hypoglycemic Agents(metformin)?

hypoglycemic Agents(metformin) is developed and marketed by First Affiliated Hospital of Wenzhou Medical University (see full First Affiliated Hospital of Wenzhou Medical University pipeline at /company/first-affiliated-hospital-of-wenzhou-medical-university).

What drug class is hypoglycemic Agents(metformin) in?

hypoglycemic Agents(metformin) belongs to the Biguanide class. See all Biguanide drugs at /class/biguanide.

What development phase is hypoglycemic Agents(metformin) in?

hypoglycemic Agents(metformin) is FDA-approved (marketed).

What are the side effects of hypoglycemic Agents(metformin)?

Common side effects of hypoglycemic Agents(metformin) include Gastrointestinal disturbance (nausea, diarrhea, abdominal discomfort), Metallic taste, Vitamin B12 deficiency, Lactic acidosis (rare, in renal impairment).

What does hypoglycemic Agents(metformin) target?

hypoglycemic Agents(metformin) targets AMP-activated protein kinase (AMPK); complex I of the mitochondrial electron transport chain and is a Biguanide.

Related

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing