Last reviewed · How we verify

HSK21542 tablet

Xizang Haisco Pharmaceutical Co., Ltd · FDA-approved active Small molecule

HSK21542 is a small-molecule inhibitor that targets specific kinases involved in cellular signaling pathways.

HSK21542 is an investigational drug developed by Xizang Haisco Pharmaceutical Co., Ltd. It is currently in Phase 2 trials for chemotherapy-induced nausea and vomiting, peritoneal dialysis pruritus, and sleep quality in hemodialysis patients with CKD-aP. The drug has not yet received FDA approval.

At a glance

Generic nameHSK21542 tablet
Also known asHSK21542, HSK21542 0.2 μg/kg, HSK21542 0.5 μg/kg, HSK21542 1 μg/kg, HSK21542 0.75 μg/kg
SponsorXizang Haisco Pharmaceutical Co., Ltd
ModalitySmall molecule
Therapeutic areaOncology
PhaseFDA-approved

Mechanism of action

While detailed mechanistic information is limited in public sources, HSK21542 appears to function as a kinase inhibitor developed for oncological applications. The drug is marketed in China by Xizang Haisco Pharmaceutical, suggesting it has completed clinical development and regulatory approval in that region.

Approved indications

No approved indications tracked.

Common side effects

No common side effects on file.

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