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Heparin or Bivalirudin

CCRF Consulting Co., Ltd. · FDA-approved active Small molecule

Heparin and bivalirudin are anticoagulants that prevent blood clot formation by inhibiting thrombin and other coagulation factors.

Heparin and bivalirudin are anticoagulants that prevent blood clot formation by inhibiting thrombin and other coagulation factors. Used for Acute coronary syndrome, Percutaneous coronary intervention, Venous thromboembolism prophylaxis and treatment.

At a glance

Generic nameHeparin or Bivalirudin
SponsorCCRF Consulting Co., Ltd.
Drug classAnticoagulant
TargetThrombin (Factor IIa) and Factor Xa (heparin); Thrombin (Factor IIa) (bivalirudin)
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Heparin is an indirect thrombin inhibitor that works through antithrombin III to inactivate factors IIa and Xa in the coagulation cascade. Bivalirudin is a direct thrombin inhibitor that binds directly to thrombin's active site and fibrin-binding site, preventing clot formation. Both are used to prevent thrombotic events in acute coronary syndromes and during percutaneous coronary intervention.

Approved indications

Common side effects

Key clinical trials

Primary sources

Every claim on this page is sourced from regulatory or scientific primary sources. See our editorial policy for full methodology.

SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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