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FOLFRINOX

Zhejiang Cancer Hospital · Phase 3 active Small molecule

FOLFRINOX is a combination chemotherapy regimen that uses multiple cytotoxic agents to inhibit DNA synthesis and cell division in cancer cells.

FOLFRINOX is a combination chemotherapy regimen that uses multiple cytotoxic agents to inhibit DNA synthesis and cell division in cancer cells. Used for Metastatic pancreatic cancer, Metastatic colorectal cancer, Gastric cancer.

At a glance

Generic nameFOLFRINOX
Also known asIrinotecan,Oxaliplatin and 5-FU
SponsorZhejiang Cancer Hospital
Drug classCombination chemotherapy regimen
ModalitySmall molecule
Therapeutic areaOncology
PhasePhase 3

Mechanism of action

FOLFRINOX combines 5-fluorouracil (5-FU), leucovorin (folinic acid), oxaliplatin, and irinotecan. 5-FU and leucovorin inhibit thymidylate synthase to disrupt DNA synthesis; oxaliplatin is a platinum agent that creates DNA crosslinks; and irinotecan inhibits topoisomerase I. Together, these agents provide synergistic cytotoxic effects against rapidly dividing cancer cells.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results